Dzina | DAPTOMYCIAN |
Nambala ya cas | 103060-53-3 |
Mawonekedwe a matope | C72h101717O26 |
Kulemera kwa maselo | 1620.67 |
Nambala ya Einecs | 600-389-2 |
Malo osungunuka | 202-204 ° C |
Malo otentha | 2078.2 ± 65.0 ° C (Zonenedweratu) |
Kukula | 1.45 ± 0,1 g / cm3 (kulosera) |
pophulikira | 87 ℃ |
Malo osungira | Osindikizidwa muuma, sitolo mu freezer, pansi -20 ° C |
Kusalola | Methanol: SoldubleG5mg / ml |
Acidity zolimba | (PKA) 4.00 ± 0,10 (ENGANI) |
Fumu | pawuda |
Mtundu | zopanda maonekedwe |
N- [[1-(1-Oxdecyl) -l-D-Asn-l ; N-[N-Decanoyll-L-D-Asn-l-asclo [a asn-l-a ask-l-a Aminobnzoyl) ecyl) -l-tryiptophyl-d-asparginyl-l-α-asnithinyl-l-α Glutamyl-α, diaminio-γ-obo-benzenebuanuadid (13-4) lactompine; diptomycin, huptomycin.
Antibiotic Diptmycin ndi a cyclipoctide antibayotic ndi gawo latsopano lomwe limatulutsidwa mu msuzi wa strummys (S. Reftospostes), zomwe zimalepheretsa bitosynthes), yomwe imalepheretsa bitosynthes Kusinthanitsa kwa membrane wa cytoplasmic kumatha kusokoneza ma bankhuni a bacrane ntchito m'njira zingapo ndikupha mabakiteriya okoma. Kuphatikiza pa kuthekera kwake kuchitira mabakiteriya okwanira kwambiri azachipatala, diptomycin ndikofunikira kwambiri kwa zovuta zakutali zomwe zawonetsa kukana methicillin, vancomycin, ndi genoczolid mu vitro. Ili ndi ntchito ya panter, ndipo malowa ali ndi tanthauzo lofunikira kwambiri azachipatala odwala. Eosinophic chibayo ndi matenda osowa komanso owopsa kwambiri ndi matendawa kuphatikizapo kutentha thupi, kutsokomola, kupuma.
Diptmycin ali ndi bacteritic yabwino kwa mabakiteriya osiyanasiyana oletsa mantififi, monga mic = 0.06-0.5 μg / ml.5 Mic = 0.0625 ~ 1μg / ml ya mabakiteriya, mic = 0.5μg / ml ya gmrbia - exaccus-exococcus ndi 0.5 ~ 1μg / ml, ndi mic of enteroclus kugonjetsedwa ndi maantibayotiki ndi 1 ~ 2μg / ml.