Tirzepatide ndi buku lodziwika bwino la insulinotropic polypeptide (GIP) lomwe limagwira ntchito pawiri la glucose komanso glucagon-like peptide-1 (GLP-1) receptor agonist. Zimayimira kupita patsogolo kwakukulu pamankhwala amtundu wa 2 shuga ndipo zawonetsa zotsatira zabwino pakuwongolera kulemera. Tirzepatide jekeseni ufa ndi mawonekedwe a mankhwala omwe amagwiritsidwa ntchito pokonzekera njira yothetsera subcutaneous administration.
Njira Yochitira
Tirzepatide imagwira ntchito poyambitsa ma GIP ndi GLP-1 receptors, omwe amawongolera kuchuluka kwa shuga m'magazi ndi chilakolako. Agonism yapawiri imapereka zotsatira zingapo zopindulitsa:
Kuchuluka kwa Insulin Katulutsidwe ka insulini: Imathandizira kutulutsidwa kwa insulin m'njira yodalira shuga, kumathandizira kutsitsa shuga wamagazi popanda kuyambitsa hypoglycemia.
Kutulutsidwa kwa Glucagon Woponderezedwa: Kumachepetsa katulutsidwe ka glucagon, timadzi timene timatulutsa shuga m'magazi.
Kuwongolera Kulakalaka: Kumalimbikitsa kukhuta ndikuchepetsa kudya, kumathandizira kuchepetsa thupi.
Kutulutsa M'mimba Mwapang'onopang'ono: Kumachedwetsa kutulutsa m'mimba, zomwe zimathandizira kuwongolera kuchuluka kwa shuga m'magazi pambuyo pakudya.
Kugwiritsa Ntchito Kovomerezeka
Monga zosintha zaposachedwa, Tirzepatide idavomerezedwa ndi olamulira monga US Food and Drug Administration (FDA) pochiza matenda amtundu wa 2. Ikufufuzidwanso kuti igwiritsidwe ntchito poyang'anira kunenepa kwambiri.
Ubwino
Kuwongolera Bwino kwa Glycemic: Kuchepetsa kwakukulu kwa milingo ya HbA1c.
Kuchepetsa Kunenepa: Kuchepetsa thupi kwambiri, komwe kumakhala kopindulitsa kwa odwala omwe ali ndi matenda amtundu wa 2 komanso kunenepa kwambiri.
Mapindu a Pamtima: Kusintha komwe kungachitike paziwopsezo zamtima, ngakhale maphunziro omwe akupitilira akuwunikanso mbali iyi.
Kusavuta: Kumwa kamodzi pamlungu kumapangitsa kuti odwala azitsatira bwino poyerekeza ndi mankhwala a tsiku ndi tsiku.
Zomwe Zingatheke
Ngakhale kuti Tirzepatide nthawi zambiri imaloledwa bwino, ogwiritsa ntchito ena amatha kukhala ndi zotsatirapo, kuphatikiza:
Mavuto a m'mimba:
Mseru, kusanza, kutsekula m'mimba, ndi kudzimbidwa ndizofala makamaka akamayamba kulandira chithandizo.
Chiwopsezo cha Hypoglycemia: Makamaka mukagwiritsidwa ntchito limodzi ndi mankhwala ena otsitsa shuga.
Pancreatitis: Chosowa koma chowopsa, chomwe chimafuna chithandizo chamankhwala mwamsanga ngati zizindikiro monga kupweteka kwa m'mimba kumachitika.
Kukonzekera ndi Kulamulira
Ufa wa jekeseni wa Tirzepatide uyenera kukonzedwanso ndi chosungunulira choyenera (kawirikawiri choperekedwa mu kit) kuti apange njira yothetsera jekeseni. Yankho lokonzedwanso liyenera kukhala lomveka bwino komanso lopanda tinthu tating'onoting'ono. Amagwiritsidwa ntchito pansi pamimba, ntchafu, kapena kumtunda kwa mkono.