Zogulitsa
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Mtengo wa CJC-1295
CJC-1295 API imapangidwa pogwiritsa ntchito ukadaulo wa solid phase peptide synthesis (SPPS) ndikuyeretsedwa pogwiritsa ntchito HPLC kuti ikwaniritse chiyero chapamwamba komanso kusasinthika kwa batch-to-batch.
Zogulitsa:Kuyera ≥ 99%
Low zotsalira zosungunulira ndi heavy metals
Endotoxin-free, non-immunogenic synthesis njira
Kuchuluka komwe mungasinthidwe: mg mpaka kg
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NAD +
Mawonekedwe a API:
Kuyera kwakukulu ≥99%
Pharmaceutical-grade NAD+
Miyezo yopanga ngati GMP
NAD+ API ndiyabwino kugwiritsidwa ntchito muzakudya zopatsa thanzi, zobaya jakisoni, komanso njira zotsogola za metabolic.
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Boc-Tyr(tBu)-Aib-Glu(OtBu)-Gly-OH
Boc-Tyr(tBu)-Aib-Glu(OtBu)-Gly-OHndi tetrapeptide yotetezedwa yomwe imagwiritsidwa ntchito pofufuza kaphatikizidwe ka peptide. Magulu a Boc (tert-butyloxycarbonyl) ndi tBu (tert-butyl) amagwira ntchito ngati magulu otchinjiriza kuti asatengere mbali pakupanga ma peptide. Kuphatikizidwa kwa Aib (α-aminoisobutyric acid) kumathandizira kupanga mapangidwe a helical ndikuwonjezera kukhazikika kwa peptide. Kutsatizana kwa peptide kumeneku kumaphunziridwa chifukwa cha kuthekera kwake pakuwunika kogwirizana, kupindika kwa peptide, komanso ngati chomangira pakupanga ma peptide a bioactive ndi kukhazikika kokhazikika komanso kukhazikika.
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Cagrilintide
Cagrilintide ndi mankhwala, amylin receptor agonist opangidwa kwa nthawi yayitali omwe amapangidwa kuti athe kuchiza kunenepa kwambiri komanso zovuta zokhudzana ndi kagayidwe kachakudya. Potengera mahomoni achilengedwe amylin, amathandizira kuwongolera njala, kuchepa kwa m'mimba, ndikuwonjezera kukhuta. API yathu yoyera kwambiri ya Cagrilintide imapangidwa pogwiritsa ntchito kaphatikizidwe kamankhwala ndipo imakwaniritsa miyezo yamagulu amankhwala, ndikupangitsa kuti ikhale yoyenera kugwiritsidwa ntchito popanga zowongolera zolemera.
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Tesamorelin
Tesamorelin API imagwiritsa ntchito ukadaulo wapamwamba kwambiri wa gawo la peptide synthesis (SPPS) ndipo ili ndi izi:
Kuyera ≥99% (HPLC)
Palibe endotoxin, zitsulo zolemera, zosungunulira zotsalira zoyesedwa
Kutsatizana kwa amino acid ndi kapangidwe kamene kamatsimikiziridwa ndi LC-MS/NMR
Perekani zopanga makonda mu magalamu mpaka ma kilogalamu -
Fmoc-Ile-Aib-OH
Fmoc-Ile-Aib-OH ndi chomangira cha dipeptide chomwe chimagwiritsidwa ntchito popanga peptide synthesis (SPPS). Zimaphatikiza Fmoc-protected isoleucine ndi Aib (α-aminoisobutyric acid), amino acid omwe si achilengedwe omwe amachititsa kuti helix ikhale yolimba komanso kukana kwa protease.
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Fmoc-L-Ls[Eic(OtBu)-γ-Glu(OtBu)-AEEA-AEEA]-OH
Fmoc-L-Lys[Eic(OtBu)-γ-Glu(OtBu)-AEEA-AEEA]-OH ndi chipika chomangira cha amino acid chomwe chimapangidwa kuti chizigwiritsidwa ntchito popereka mankhwala ndi bioconjugation. Imakhala ndi gawo la Eic (eicosanoid) lolumikizana ndi lipid, γ-Glu polunjika, ndi ma spacers a AEEA kuti athe kusinthasintha.
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Boc-Tyr(tBu)-Aib-OH
Boc-Tyr(tBu)-Aib-OH ndi chomangira chotetezedwa cha dipeptide chomwe chimagwiritsidwa ntchito popanga peptide, kuphatikiza Boc-protected tyrosine ndi Aib (α-aminoisobutyric acid). Zotsalira za Aib zimakulitsa mapangidwe a helix ndi kukana kwa protease.
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Boc-His(Trt)-Ala-Glu(OtBu)-Gly-OH
Boc-His(Trt)-Ala-Glu(OtBu)-Gly-OH ndi chidutswa chotetezedwa cha tetrapeptide chomwe chimagwiritsidwa ntchito popanga peptide synthesis (SPPS) ndi chitukuko cha mankhwala a peptide. Zimaphatikizapo magulu otetezera a orthogonal synthesis ndipo imakhala ndi ndondomeko yothandiza pakupanga mapangidwe a peptide.
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Fmoc-Ls(Pal-Glu-OtBu)-OH
Fmoc-Ls(Pal-Glu-OtBu) -OH ndi chipika chapadera cha amino acid chomangira chopangira peptide-lipid conjugation. Imakhala ndi lysine yotetezedwa ndi Fmoc yokhala ndi unyolo wam'mbali wa palmitoyl-glutamate, kukulitsa kuyanjana kwa membrane ndi bioavailability.
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Fmoc-His-Aib-OH
Fmoc-His-Aib-OH ndi chomangira cha dipeptide chomwe chimagwiritsidwa ntchito popanga peptide, kuphatikiza Fmoc-protected histidine ndi Aib (α-aminoisobutyric acid). Aib imayambitsa kukhazikika kwa conformational, ndikupangitsa kuti ikhale yofunikira popanga ma helical ndi okhazikika ma peptides.
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Boc-His(Trt)-Aib-Glu(OtBu)-Gly-OH
Boc-His(Trt)-Aib-Glu(OtBu)-Gly-OH ndi chidutswa chotetezedwa cha tetrapeptide chomwe chimagwiritsidwa ntchito popanga peptide ndi chitukuko cha mankhwala. Lili ndi magulu ogwira ntchito otetezedwa mwanzeru kuti agwirizane pang'onopang'ono komanso amakhala ndi Aib (α-aminoisobutyric acid) kuti apititse patsogolo kukhazikika kwa helix ndi kukhazikika kogwirizana.
