Melanotan 1ndi synthetic peptide analogue ofα-MSH (mahomoni olimbikitsa alpha-melanocyte). Imagwira ntchito ndikuyambitsa melanocortin-1 receptors (MC1R)kulimbikitsakupanga melanin, kupereka zachilengedwekhungu la pigmentationndiPhotoprotection.
Zinalizovomerezeka zochizira erythropoietic protoporphyria (EPP)-matenda osowa omwe amachititsa kumva kwambiri ndi kuwala kwa dzuwa. Melanotan 1 imathandizira kuwonjezekakulekerera kwa UV kuwala, kuchepetsazotsatira za phototoxic, ndi kuwonjezerachitetezo cha khungu ku kuwonongeka kwa UV.
ZosankhaChithunzi cha MC1R
Kuwonjezekakupanga eumelanin
Amaperekachitetezo chachilengedwe cha dzuwa
ImathandiziraDNA kukonza ndi kuyankha odana ndi kutupa
Zotheka zavitiligo, kupewa khansa yapakhungu,ndizodzikongoletsera pigmentation
Kufufuzidwa muanti-kukalambandidermatological mankhwala
Kuyera kwakukulu ≥99%
Solid-phase peptide synthesis (SPPS)
Miyezo yopanga ngati GMP
Kupezeka kochulukira: R&D mpaka magawo azamalonda